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氟马西尼

英文名: flumazenil

CAS: 78755-81-4      分子式: C15H14FN3O3

分子量: 303.28800

别名:


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描述

Flumazenil (also known as flumazepil, code name Ro 15-1788) is a selective benzodiazepine receptor antagonist primarily available by injection only, and the only GABAA negative allosteric modulator on the market today. It has antagonistic and antidote properties to therapeutically used benzodiazapenes, through competitive inhibition. It was first introduced in 1987 by Hoffmann-La Roche under the trade name Anexate, but only approved by the FDA on December 20, 1991. Flumazenil went off patent in 2008 so at present generic formulations of this drug are available. Intravenous flumazenil is primarily used to treat benzodiazepine overdoses and to help reverse anesthesia. Administration of flumazenil by sublingual lozenge and topical cream has also been tested.

基本信息
英文名:
flumazenil
CAS号.:
78755-81-4
别名:
YM-684; RO 15-1788; Romazicon; Mazicon; Flumazepil; Lanexat; ANEXATE; Flumazenil; FMZ; Ro 1722;
分子式:
C15H14FN3O3
分子量:
303.28800
PSA:
64.43000
LogP:
1.71160
物化属性
外观:
密度:
熔点:
201-203°C
沸点:
闪点:
储存条件:
2-8°C
安全信息
海关编码:
2933990090
WGK Germany:
2
危险类别码:
R36/37/38
安全说明:
S26; S27; S36/37/39
危险品标志:
Xi
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